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    <link:label id="lab_exel_BuiltToSuitLeaseMember_75B7CDA49781D18A2B0B0FD638A8535C_terseLabel_en-US" xlink:label="lab_exel_BuiltToSuitLeaseMember_75B7CDA49781D18A2B0B0FD638A8535C" xlink:role="http://www.xbrl.org/2003/role/terseLabel" xlink:type="resource" xml:lang="en-US">Built-To-Suit Lease</link:label>
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    <link:label id="lab_srt_StatementGeographicalAxis_3A2F9F645B7AB022985F0F9CE26EDB0E_label_en-US" xlink:label="lab_srt_StatementGeographicalAxis_3A2F9F645B7AB022985F0F9CE26EDB0E" xlink:role="http://www.xbrl.org/2003/role/label" xlink:type="resource" xml:lang="en-US">Geographical [Axis]</link:label>
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    <link:label id="lab_srt_SegmentGeographicalDomain_F97437AD679F0AC7A0FF0F9CE26E2504_terseLabel_en-US" xlink:label="lab_srt_SegmentGeographicalDomain_F97437AD679F0AC7A0FF0F9CE26E2504" xlink:role="http://www.xbrl.org/2003/role/terseLabel" xlink:type="resource" xml:lang="en-US">Geographical [Domain]</link:label>
    <link:label id="lab_srt_SegmentGeographicalDomain_F97437AD679F0AC7A0FF0F9CE26E2504_label_en-US" xlink:label="lab_srt_SegmentGeographicalDomain_F97437AD679F0AC7A0FF0F9CE26E2504" xlink:role="http://www.xbrl.org/2003/role/label" xlink:type="resource" xml:lang="en-US">Geographical [Domain]</link:label>
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    <link:label id="lab_us-gaap_SubsequentEventLineItems_472BA4E1FFA9733CA93D0F9CE2700A10_terseLabel_en-US" xlink:label="lab_us-gaap_SubsequentEventLineItems_472BA4E1FFA9733CA93D0F9CE2700A10" xlink:role="http://www.xbrl.org/2003/role/terseLabel" xlink:type="resource" xml:lang="en-US">Subsequent Event [Line Items]</link:label>
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    <link:label id="lab_us-gaap_AreaOfRealEstateProperty_A23D7A095B13A28537160F9CE270E573_terseLabel_en-US" xlink:label="lab_us-gaap_AreaOfRealEstateProperty_A23D7A095B13A28537160F9CE270E573" xlink:role="http://www.xbrl.org/2003/role/terseLabel" xlink:type="resource" xml:lang="en-US">Area of lease property (in square feet)</link:label>
    <link:label id="lab_us-gaap_AreaOfRealEstateProperty_A23D7A095B13A28537160F9CE270E573_label_en-US" xlink:label="lab_us-gaap_AreaOfRealEstateProperty_A23D7A095B13A28537160F9CE270E573" xlink:role="http://www.xbrl.org/2003/role/label" xlink:type="resource" xml:lang="en-US">Area of Real Estate Property</link:label>
    <link:loc xlink:href="http://xbrl.fasb.org/us-gaap/2019/elts/us-gaap-2019-01-31.xsd#us-gaap_AreaOfRealEstateProperty" xlink:label="loc_us-gaap_AreaOfRealEstateProperty_A23D7A095B13A28537160F9CE270E573" xlink:type="locator" />
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    <link:label id="lab_us-gaap_LesseeOperatingLeaseTermOfContract_BB1DC71E62A3154AA4510F9CE2704AD4_terseLabel_en-US" xlink:label="lab_us-gaap_LesseeOperatingLeaseTermOfContract_BB1DC71E62A3154AA4510F9CE2704AD4" xlink:role="http://www.xbrl.org/2003/role/terseLabel" xlink:type="resource" xml:lang="en-US">Operating lease term</link:label>
    <link:label id="lab_us-gaap_LesseeOperatingLeaseTermOfContract_BB1DC71E62A3154AA4510F9CE2704AD4_label_en-US" xlink:label="lab_us-gaap_LesseeOperatingLeaseTermOfContract_BB1DC71E62A3154AA4510F9CE2704AD4" xlink:role="http://www.xbrl.org/2003/role/label" xlink:type="resource" xml:lang="en-US">Lessee, Operating Lease, Term of Contract</link:label>
    <link:loc xlink:href="http://xbrl.fasb.org/us-gaap/2019/elts/us-gaap-2019-01-31.xsd#us-gaap_LesseeOperatingLeaseTermOfContract" xlink:label="loc_us-gaap_LesseeOperatingLeaseTermOfContract_BB1DC71E62A3154AA4510F9CE2704AD4" xlink:type="locator" />
    <link:labelArc order="1" xlink:arcrole="http://www.xbrl.org/2003/arcrole/concept-label" xlink:from="loc_us-gaap_LesseeOperatingLeaseTermOfContract_BB1DC71E62A3154AA4510F9CE2704AD4" xlink:to="lab_us-gaap_LesseeOperatingLeaseTermOfContract_BB1DC71E62A3154AA4510F9CE2704AD4" xlink:type="arc" />
    <link:label id="lab_exel_LesseeOperatingLeaseNotYetCommencedMonthlyBasePayment_D8AACE7C210665FD1BB90F9CE270C18D_terseLabel_en-US" xlink:label="lab_exel_LesseeOperatingLeaseNotYetCommencedMonthlyBasePayment_D8AACE7C210665FD1BB90F9CE270C18D" xlink:role="http://www.xbrl.org/2003/role/terseLabel" xlink:type="resource" xml:lang="en-US">Estimated monthly base rent under Build-to-Suite Leases</link:label>
    <link:label id="lab_exel_LesseeOperatingLeaseNotYetCommencedMonthlyBasePayment_D8AACE7C210665FD1BB90F9CE270C18D_label_en-US" xlink:label="lab_exel_LesseeOperatingLeaseNotYetCommencedMonthlyBasePayment_D8AACE7C210665FD1BB90F9CE270C18D" xlink:role="http://www.xbrl.org/2003/role/label" xlink:type="resource" xml:lang="en-US">Lessee, Operating Lease, Not Yet Commenced, Monthly Base Payment</link:label>
    <link:label id="lab_exel_LesseeOperatingLeaseNotYetCommencedMonthlyBasePayment_D8AACE7C210665FD1BB90F9CE270C18D_documentation_en-US" xlink:label="lab_exel_LesseeOperatingLeaseNotYetCommencedMonthlyBasePayment_D8AACE7C210665FD1BB90F9CE270C18D" xlink:role="http://www.xbrl.org/2003/role/documentation" xlink:type="resource" xml:lang="en-US">Lessee, Operating Lease, Not Yet Commenced, Monthly Base Payment</link:label>
    <link:loc xlink:href="exel-20190927.xsd#exel_LesseeOperatingLeaseNotYetCommencedMonthlyBasePayment" xlink:label="loc_exel_LesseeOperatingLeaseNotYetCommencedMonthlyBasePayment_D8AACE7C210665FD1BB90F9CE270C18D" xlink:type="locator" />
    <link:labelArc order="1" xlink:arcrole="http://www.xbrl.org/2003/arcrole/concept-label" xlink:from="loc_exel_LesseeOperatingLeaseNotYetCommencedMonthlyBasePayment_D8AACE7C210665FD1BB90F9CE270C18D" xlink:to="lab_exel_LesseeOperatingLeaseNotYetCommencedMonthlyBasePayment_D8AACE7C210665FD1BB90F9CE270C18D" xlink:type="arc" />
    <link:label id="lab_exel_LesseeOperatingLeaseNotYetCommencedMonthlyBasePaymentAnnualIncreasePercentage_B1FC945D988EA6F5CD140F9CE2705A1A_terseLabel_en-US" xlink:label="lab_exel_LesseeOperatingLeaseNotYetCommencedMonthlyBasePaymentAnnualIncreasePercentage_B1FC945D988EA6F5CD140F9CE2705A1A" xlink:role="http://www.xbrl.org/2003/role/terseLabel" xlink:type="resource" xml:lang="en-US">Monthly base rent, lease not yet commenced, annual percentage increase</link:label>
    <link:label id="lab_exel_LesseeOperatingLeaseNotYetCommencedMonthlyBasePaymentAnnualIncreasePercentage_B1FC945D988EA6F5CD140F9CE2705A1A_label_en-US" xlink:label="lab_exel_LesseeOperatingLeaseNotYetCommencedMonthlyBasePaymentAnnualIncreasePercentage_B1FC945D988EA6F5CD140F9CE2705A1A" xlink:role="http://www.xbrl.org/2003/role/label" xlink:type="resource" xml:lang="en-US">Lessee, Operating Lease, Not Yet Commenced, Monthly Base Payment, Annual Increase, Percentage</link:label>
    <link:label id="lab_exel_LesseeOperatingLeaseNotYetCommencedMonthlyBasePaymentAnnualIncreasePercentage_B1FC945D988EA6F5CD140F9CE2705A1A_documentation_en-US" xlink:label="lab_exel_LesseeOperatingLeaseNotYetCommencedMonthlyBasePaymentAnnualIncreasePercentage_B1FC945D988EA6F5CD140F9CE2705A1A" xlink:role="http://www.xbrl.org/2003/role/documentation" xlink:type="resource" xml:lang="en-US">Lessee, Operating Lease, Not Yet Commenced, Monthly Base Payment, Annual Increase, Percentage</link:label>
    <link:loc xlink:href="exel-20190927.xsd#exel_LesseeOperatingLeaseNotYetCommencedMonthlyBasePaymentAnnualIncreasePercentage" xlink:label="loc_exel_LesseeOperatingLeaseNotYetCommencedMonthlyBasePaymentAnnualIncreasePercentage_B1FC945D988EA6F5CD140F9CE2705A1A" xlink:type="locator" />
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    <link:label id="lab_exel_LesseeOperatingLeaseNumberOfRenewalOptions_A70AB0F9F0C0B97726EB0F9CE270FF8C_terseLabel_en-US" xlink:label="lab_exel_LesseeOperatingLeaseNumberOfRenewalOptions_A70AB0F9F0C0B97726EB0F9CE270FF8C" xlink:role="http://www.xbrl.org/2003/role/terseLabel" xlink:type="resource" xml:lang="en-US">Number of options to extend the Lease</link:label>
    <link:label id="lab_exel_LesseeOperatingLeaseNumberOfRenewalOptions_A70AB0F9F0C0B97726EB0F9CE270FF8C_label_en-US" xlink:label="lab_exel_LesseeOperatingLeaseNumberOfRenewalOptions_A70AB0F9F0C0B97726EB0F9CE270FF8C" xlink:role="http://www.xbrl.org/2003/role/label" xlink:type="resource" xml:lang="en-US">Lessee, Operating Lease, Number Of Renewal Options</link:label>
    <link:label id="lab_exel_LesseeOperatingLeaseNumberOfRenewalOptions_A70AB0F9F0C0B97726EB0F9CE270FF8C_documentation_en-US" xlink:label="lab_exel_LesseeOperatingLeaseNumberOfRenewalOptions_A70AB0F9F0C0B97726EB0F9CE270FF8C" xlink:role="http://www.xbrl.org/2003/role/documentation" xlink:type="resource" xml:lang="en-US">Lessee, Operating Lease, Number Of Renewal Options</link:label>
    <link:loc xlink:href="exel-20190927.xsd#exel_LesseeOperatingLeaseNumberOfRenewalOptions" xlink:label="loc_exel_LesseeOperatingLeaseNumberOfRenewalOptions_A70AB0F9F0C0B97726EB0F9CE270FF8C" xlink:type="locator" />
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    <link:label id="lab_us-gaap_LesseeOperatingLeaseRenewalTerm_F4556FACCB2A7433C5860FCB7778FD31_terseLabel_en-US" xlink:label="lab_us-gaap_LesseeOperatingLeaseRenewalTerm_F4556FACCB2A7433C5860FCB7778FD31" xlink:role="http://www.xbrl.org/2003/role/terseLabel" xlink:type="resource" xml:lang="en-US">Lease option to extend period</link:label>
    <link:label id="lab_us-gaap_LesseeOperatingLeaseRenewalTerm_F4556FACCB2A7433C5860FCB7778FD31_label_en-US" xlink:label="lab_us-gaap_LesseeOperatingLeaseRenewalTerm_F4556FACCB2A7433C5860FCB7778FD31" xlink:role="http://www.xbrl.org/2003/role/label" xlink:type="resource" xml:lang="en-US">Lessee, Operating Lease, Renewal Term</link:label>
    <link:loc xlink:href="http://xbrl.fasb.org/us-gaap/2019/elts/us-gaap-2019-01-31.xsd#us-gaap_LesseeOperatingLeaseRenewalTerm" xlink:label="loc_us-gaap_LesseeOperatingLeaseRenewalTerm_F4556FACCB2A7433C5860FCB7778FD31" xlink:type="locator" />
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    <link:label id="lab_exel_LesseeOperatingLeaseOptionToTerminateAfterPeriod_0CF7CF5B7DFCE5C36D9C0FD4B1D6B14F_terseLabel_en-US" xlink:label="lab_exel_LesseeOperatingLeaseOptionToTerminateAfterPeriod_0CF7CF5B7DFCE5C36D9C0FD4B1D6B14F" xlink:role="http://www.xbrl.org/2003/role/terseLabel" xlink:type="resource" xml:lang="en-US">Option to terminate lease (after period)</link:label>
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    <link:label id="lab_exel_OperatingLeaseAdditionalAreaOfRealEstateProperty_0E90C56871C6A7D60F5C0FDE6E16AA18_terseLabel_en-US" xlink:label="lab_exel_OperatingLeaseAdditionalAreaOfRealEstateProperty_0E90C56871C6A7D60F5C0FDE6E16AA18" xlink:role="http://www.xbrl.org/2003/role/terseLabel" xlink:type="resource" xml:lang="en-US">Operating lease, expansion (in square feet)</link:label>
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    <link:label id="lab_us-gaap_BalanceSheetLocationDomain_75223321FA17AEA24E38E31EA0AD8D3D_label_en-US" xlink:label="lab_us-gaap_BalanceSheetLocationDomain_5D22FEBE209A54558023752CEDF917C6" xlink:role="http://www.xbrl.org/2003/role/label" xlink:type="resource" xml:lang="en-US">Balance Sheet Location [Domain]</link:label>
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    <link:label id="lab_us-gaap_InventoriesMember_403A904ABB913EE84C93E31EA0AE7D21_terseLabel_en-US" xlink:label="lab_us-gaap_InventoriesMember_E31F1D02E99B5F279E654FB968F68F51" xlink:role="http://www.xbrl.org/2003/role/terseLabel" xlink:type="resource" xml:lang="en-US">Current portion included in Inventory</link:label>
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    <link:loc xlink:href="http://xbrl.fasb.org/us-gaap/2019/elts/us-gaap-2019-01-31.xsd#us-gaap_IncreaseDecreaseInEmployeeRelatedLiabilities" xlink:label="loc_us-gaap_IncreaseDecreaseInEmployeeRelatedLiabilities_226E8BFFFF849A7BB9EE199E158406F5" xlink:type="locator" />
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    <link:label id="lab_exel_IncreaseDecreaseInAccruedClinicalLiabilities_31F60ED1C757CE7A2D17199E15848513_terseLabel_en-US" xlink:label="lab_exel_IncreaseDecreaseInAccruedClinicalLiabilities_31F60ED1C757CE7A2D17199E15848513" xlink:role="http://www.xbrl.org/2003/role/terseLabel" xlink:type="resource" xml:lang="en-US">Accrued clinical trial liabilities</link:label>
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    <link:label id="lab_exel_IncreaseDecreaseInRebatesAndFeesPayable_93CC63D5B90017D7EFEA199E1584F51E_terseLabel_en-US" xlink:label="lab_exel_IncreaseDecreaseInRebatesAndFeesPayable_93CC63D5B90017D7EFEA199E1584F51E" xlink:role="http://www.xbrl.org/2003/role/terseLabel" xlink:type="resource" xml:lang="en-US">Rebates and fees due customers</link:label>
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    <link:label id="lab_exel_IncreaseDecreaseInRebatesAndFeesPayable_93CC63D5B90017D7EFEA199E1584F51E_documentation_en-US" xlink:label="lab_exel_IncreaseDecreaseInRebatesAndFeesPayable_93CC63D5B90017D7EFEA199E1584F51E" xlink:role="http://www.xbrl.org/2003/role/documentation" xlink:type="resource" xml:lang="en-US">Increase (Decrease) In Rebates And Fees Payable</link:label>
    <link:loc xlink:href="exel-20190927.xsd#exel_IncreaseDecreaseInRebatesAndFeesPayable" xlink:label="loc_exel_IncreaseDecreaseInRebatesAndFeesPayable_93CC63D5B90017D7EFEA199E1584F51E" xlink:type="locator" />
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    <link:label id="lab_exel_IncreaseDecreaseInAccruedCollaborationLiability_D2C3781BEE878FC037C1199E1584951F_terseLabel_en-US" xlink:label="lab_exel_IncreaseDecreaseInAccruedCollaborationLiability_D2C3781BEE878FC037C1199E1584951F" xlink:role="http://www.xbrl.org/2003/role/terseLabel" xlink:type="resource" xml:lang="en-US">Accrued collaboration liability</link:label>
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    <link:label id="lab_exel_IncreaseDecreaseInAccruedCollaborationLiability_D2C3781BEE878FC037C1199E1584951F_documentation_en-US" xlink:label="lab_exel_IncreaseDecreaseInAccruedCollaborationLiability_D2C3781BEE878FC037C1199E1584951F" xlink:role="http://www.xbrl.org/2003/role/documentation" xlink:type="resource" xml:lang="en-US">Increase (Decrease) in Accrued Collaboration Liability</link:label>
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    <link:loc xlink:href="http://xbrl.fasb.org/us-gaap/2019/elts/us-gaap-2019-01-31.xsd#us-gaap_IncreaseDecreaseInContractWithCustomerLiability" xlink:label="loc_us-gaap_IncreaseDecreaseInContractWithCustomerLiability_798939168D178572FDD0199E1584D208" xlink:type="locator" />
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    <link:label id="lab_exel_IncreaseDecreaseInLeaseLiabilityNoncurrent_23EE4479CDB2455DF0E7199E1584C815_terseLabel_en-US" xlink:label="lab_exel_IncreaseDecreaseInLeaseLiabilityNoncurrent_23EE4479CDB2455DF0E7199E1584C815" xlink:role="http://www.xbrl.org/2003/role/terseLabel" xlink:type="resource" xml:lang="en-US">Long-term portion of lease liabilities</link:label>
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    <link:label id="lab_exel_IncreaseDecreaseInLeaseLiabilityNoncurrent_23EE4479CDB2455DF0E7199E1584C815_documentation_en-US" xlink:label="lab_exel_IncreaseDecreaseInLeaseLiabilityNoncurrent_23EE4479CDB2455DF0E7199E1584C815" xlink:role="http://www.xbrl.org/2003/role/documentation" xlink:type="resource" xml:lang="en-US">Increase (Decrease) In Lease Liability, Noncurrent</link:label>
    <link:loc xlink:href="exel-20190927.xsd#exel_IncreaseDecreaseInLeaseLiabilityNoncurrent" xlink:label="loc_exel_IncreaseDecreaseInLeaseLiabilityNoncurrent_23EE4479CDB2455DF0E7199E1584C815" xlink:type="locator" />
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    <link:label id="lab_us-gaap_IncreaseDecreaseInOtherOperatingLiabilities_35828C7343ED34AB1FF1199E158485F3_terseLabel_en-US" xlink:label="lab_us-gaap_IncreaseDecreaseInOtherOperatingLiabilities_35828C7343ED34AB1FF1199E158485F3" xlink:role="http://www.xbrl.org/2003/role/terseLabel" xlink:type="resource" xml:lang="en-US">Other current and long-term liabilities</link:label>
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    <link:loc xlink:href="http://xbrl.fasb.org/us-gaap/2019/elts/us-gaap-2019-01-31.xsd#us-gaap_IncreaseDecreaseInOtherOperatingLiabilities" xlink:label="loc_us-gaap_IncreaseDecreaseInOtherOperatingLiabilities_35828C7343ED34AB1FF1199E158485F3" xlink:type="locator" />
    <link:labelArc order="1" xlink:arcrole="http://www.xbrl.org/2003/arcrole/concept-label" xlink:from="loc_us-gaap_IncreaseDecreaseInOtherOperatingLiabilities_35828C7343ED34AB1FF1199E158485F3" xlink:to="lab_us-gaap_IncreaseDecreaseInOtherOperatingLiabilities_35828C7343ED34AB1FF1199E158485F3" xlink:type="arc" />
    <link:label id="lab_us-gaap_NetCashProvidedByUsedInOperatingActivities_6C19D505A73C50FD3DBF199E15851384_totalLabel_en-US" xlink:label="lab_us-gaap_NetCashProvidedByUsedInOperatingActivities_6C19D505A73C50FD3DBF199E15851384" xlink:role="http://www.xbrl.org/2003/role/totalLabel" xlink:type="resource" xml:lang="en-US">Net cash provided by operating activities</link:label>
    <link:label id="lab_us-gaap_NetCashProvidedByUsedInOperatingActivities_6C19D505A73C50FD3DBF199E15851384_label_en-US" xlink:label="lab_us-gaap_NetCashProvidedByUsedInOperatingActivities_6C19D505A73C50FD3DBF199E15851384" xlink:role="http://www.xbrl.org/2003/role/label" xlink:type="resource" xml:lang="en-US">Net Cash Provided by (Used in) Operating Activities</link:label>
    <link:loc xlink:href="http://xbrl.fasb.org/us-gaap/2019/elts/us-gaap-2019-01-31.xsd#us-gaap_NetCashProvidedByUsedInOperatingActivities" xlink:label="loc_us-gaap_NetCashProvidedByUsedInOperatingActivities_6C19D505A73C50FD3DBF199E15851384" xlink:type="locator" />
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    <link:label id="lab_us-gaap_NetCashProvidedByUsedInInvestingActivitiesAbstract_6AAE2A9E65BE76422A7E199E1585A3F6_terseLabel_en-US" xlink:label="lab_us-gaap_NetCashProvidedByUsedInInvestingActivitiesAbstract_6AAE2A9E65BE76422A7E199E1585A3F6" xlink:role="http://www.xbrl.org/2003/role/terseLabel" xlink:type="resource" xml:lang="en-US">Cash flows from investing activities:</link:label>
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    <link:label id="lab_us-gaap_PaymentsToAcquirePropertyPlantAndEquipment_11F2AC1FE3AEE27FF7FC199E158570DF_negatedLabel_en-US" xlink:label="lab_us-gaap_PaymentsToAcquirePropertyPlantAndEquipment_11F2AC1FE3AEE27FF7FC199E158570DF" xlink:role="http://www.xbrl.org/2009/role/negatedLabel" xlink:type="resource" xml:lang="en-US">Purchases of property and equipment</link:label>
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    <link:loc xlink:href="http://xbrl.fasb.org/us-gaap/2019/elts/us-gaap-2019-01-31.xsd#us-gaap_PaymentsToAcquirePropertyPlantAndEquipment" xlink:label="loc_us-gaap_PaymentsToAcquirePropertyPlantAndEquipment_11F2AC1FE3AEE27FF7FC199E158570DF" xlink:type="locator" />
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    <link:label id="lab_exel_ComputerEquipmentAndSoftwareMember_FB1017B00A9D40D5B295E23266A41A30_terseLabel_en-US" xlink:label="lab_exel_ComputerEquipmentAndSoftwareMember_07BCA2E2F43C534A858B50DD23161935" xlink:role="http://www.xbrl.org/2003/role/terseLabel" xlink:type="resource" xml:lang="en-US">Computer equipment and software</link:label>
    <link:label id="lab_exel_ComputerEquipmentAndSoftwareMember_FB1017B00A9D40D5B295E23266A41A30_label_en-US" xlink:label="lab_exel_ComputerEquipmentAndSoftwareMember_07BCA2E2F43C534A858B50DD23161935" xlink:role="http://www.xbrl.org/2003/role/label" xlink:type="resource" xml:lang="en-US">Computer Equipment And Software [Member]</link:label>
    <link:label id="lab_exel_ComputerEquipmentAndSoftwareMember_FB1017B00A9D40D5B295E23266A41A30_documentation_en-US" xlink:label="lab_exel_ComputerEquipmentAndSoftwareMember_07BCA2E2F43C534A858B50DD23161935" xlink:role="http://www.xbrl.org/2003/role/documentation" xlink:type="resource" xml:lang="en-US">Computer Equipment And Software [Member].</link:label>
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    <link:labelArc order="1" xlink:arcrole="http://www.xbrl.org/2003/arcrole/concept-label" xlink:from="loc_exel_ComputerEquipmentAndSoftwareMember_07BCA2E2F43C534A858B50DD23161935" xlink:to="lab_exel_ComputerEquipmentAndSoftwareMember_07BCA2E2F43C534A858B50DD23161935" xlink:type="arc" />
    <link:label id="lab_us-gaap_FurnitureAndFixturesMember_885BF729AC91B3CC6035E23266A4D0D5_terseLabel_en-US" xlink:label="lab_us-gaap_FurnitureAndFixturesMember_FA6D83194E17502998A59CE891201747" xlink:role="http://www.xbrl.org/2003/role/terseLabel" xlink:type="resource" xml:lang="en-US">Furniture and fixtures</link:label>
    <link:label id="lab_us-gaap_FurnitureAndFixturesMember_885BF729AC91B3CC6035E23266A4D0D5_label_en-US" xlink:label="lab_us-gaap_FurnitureAndFixturesMember_FA6D83194E17502998A59CE891201747" xlink:role="http://www.xbrl.org/2003/role/label" xlink:type="resource" xml:lang="en-US">Furniture and Fixtures [Member]</link:label>
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    <link:label id="lab_exel_LaboratoryEquipmentMember_E26806020AA1BB8014BFE23266A5EEC0_terseLabel_en-US" xlink:label="lab_exel_LaboratoryEquipmentMember_FD11A9FABE65513FB8BE2AD67FF99F50" xlink:role="http://www.xbrl.org/2003/role/terseLabel" xlink:type="resource" xml:lang="en-US">Laboratory equipment</link:label>
    <link:label id="lab_exel_LaboratoryEquipmentMember_E26806020AA1BB8014BFE23266A5EEC0_label_en-US" xlink:label="lab_exel_LaboratoryEquipmentMember_FD11A9FABE65513FB8BE2AD67FF99F50" xlink:role="http://www.xbrl.org/2003/role/label" xlink:type="resource" xml:lang="en-US">Laboratory Equipment [Member]</link:label>
    <link:label id="lab_exel_LaboratoryEquipmentMember_E26806020AA1BB8014BFE23266A5EEC0_documentation_en-US" xlink:label="lab_exel_LaboratoryEquipmentMember_FD11A9FABE65513FB8BE2AD67FF99F50" xlink:role="http://www.xbrl.org/2003/role/documentation" xlink:type="resource" xml:lang="en-US">Laboratory Equipment [Member]</link:label>
    <link:loc xlink:href="exel-20190927.xsd#exel_LaboratoryEquipmentMember" xlink:label="loc_exel_LaboratoryEquipmentMember_FD11A9FABE65513FB8BE2AD67FF99F50" xlink:type="locator" />
    <link:labelArc order="1" xlink:arcrole="http://www.xbrl.org/2003/arcrole/concept-label" xlink:from="loc_exel_LaboratoryEquipmentMember_FD11A9FABE65513FB8BE2AD67FF99F50" xlink:to="lab_exel_LaboratoryEquipmentMember_FD11A9FABE65513FB8BE2AD67FF99F50" xlink:type="arc" />
    <link:label id="lab_us-gaap_ConstructionInProgressMember_4E2DC5D6998A291A04CDE23266A5E363_terseLabel_en-US" xlink:label="lab_us-gaap_ConstructionInProgressMember_595960FA46955FFD9DA19F31C1BC41C1" xlink:role="http://www.xbrl.org/2003/role/terseLabel" xlink:type="resource" xml:lang="en-US">Construction in progress</link:label>
    <link:label id="lab_us-gaap_ConstructionInProgressMember_4E2DC5D6998A291A04CDE23266A5E363_label_en-US" xlink:label="lab_us-gaap_ConstructionInProgressMember_595960FA46955FFD9DA19F31C1BC41C1" xlink:role="http://www.xbrl.org/2003/role/label" xlink:type="resource" xml:lang="en-US">Construction in Progress [Member]</link:label>
    <link:loc xlink:href="http://xbrl.fasb.org/us-gaap/2019/elts/us-gaap-2019-01-31.xsd#us-gaap_ConstructionInProgressMember" xlink:label="loc_us-gaap_ConstructionInProgressMember_595960FA46955FFD9DA19F31C1BC41C1" xlink:type="locator" />
    <link:labelArc order="1" xlink:arcrole="http://www.xbrl.org/2003/arcrole/concept-label" xlink:from="loc_us-gaap_ConstructionInProgressMember_595960FA46955FFD9DA19F31C1BC41C1" xlink:to="lab_us-gaap_ConstructionInProgressMember_595960FA46955FFD9DA19F31C1BC41C1" xlink:type="arc" />
    <link:label id="lab_us-gaap_PropertyPlantAndEquipmentLineItems_06325C59D7D553503C7BE23266A5048C_terseLabel_en-US" xlink:label="lab_us-gaap_PropertyPlantAndEquipmentLineItems_A95B0256D7A75AF28E28518CA0A3B653" xlink:role="http://www.xbrl.org/2003/role/terseLabel" xlink:type="resource" xml:lang="en-US">Property, Plant and Equipment [Line Items]</link:label>
    <link:label id="lab_us-gaap_PropertyPlantAndEquipmentLineItems_06325C59D7D553503C7BE23266A5048C_label_en-US" xlink:label="lab_us-gaap_PropertyPlantAndEquipmentLineItems_A95B0256D7A75AF28E28518CA0A3B653" xlink:role="http://www.xbrl.org/2003/role/label" xlink:type="resource" xml:lang="en-US">Property, Plant and Equipment [Line Items]</link:label>
    <link:loc xlink:href="http://xbrl.fasb.org/us-gaap/2019/elts/us-gaap-2019-01-31.xsd#us-gaap_PropertyPlantAndEquipmentLineItems" xlink:label="loc_us-gaap_PropertyPlantAndEquipmentLineItems_A95B0256D7A75AF28E28518CA0A3B653" xlink:type="locator" />
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    <link:label id="lab_us-gaap_PropertyPlantAndEquipmentGross_6B965C8D8CC49C58D24FE23266A5A22E_terseLabel_en-US" xlink:label="lab_us-gaap_PropertyPlantAndEquipmentGross_57544161E0BB58CC97E5140A97003D1E" xlink:role="http://www.xbrl.org/2003/role/terseLabel" xlink:type="resource" xml:lang="en-US">Property and equipment, gross</link:label>
    <link:label id="lab_us-gaap_PropertyPlantAndEquipmentGross_6B965C8D8CC49C58D24FE23266A5A22E_label_en-US" xlink:label="lab_us-gaap_PropertyPlantAndEquipmentGross_57544161E0BB58CC97E5140A97003D1E" xlink:role="http://www.xbrl.org/2003/role/label" xlink:type="resource" xml:lang="en-US">Property, Plant and Equipment, Gross</link:label>
    <link:loc xlink:href="http://xbrl.fasb.org/us-gaap/2019/elts/us-gaap-2019-01-31.xsd#us-gaap_PropertyPlantAndEquipmentGross" xlink:label="loc_us-gaap_PropertyPlantAndEquipmentGross_57544161E0BB58CC97E5140A97003D1E" xlink:type="locator" />
    <link:labelArc order="1" xlink:arcrole="http://www.xbrl.org/2003/arcrole/concept-label" xlink:from="loc_us-gaap_PropertyPlantAndEquipmentGross_57544161E0BB58CC97E5140A97003D1E" xlink:to="lab_us-gaap_PropertyPlantAndEquipmentGross_57544161E0BB58CC97E5140A97003D1E" xlink:type="arc" />
    <link:label id="lab_us-gaap_AccumulatedDepreciationDepletionAndAmortizationPropertyPlantAndEquipment_69D7530A8060BB16E9ACE23266A6C0E4_negatedLabel_en-US" xlink:label="lab_us-gaap_AccumulatedDepreciationDepletionAndAmortizationPropertyPlantAndEquipment_8E93F2D3893952A7A035AC78B1D7F650" xlink:role="http://www.xbrl.org/2009/role/negatedLabel" xlink:type="resource" xml:lang="en-US">Less: accumulated depreciation and amortization</link:label>
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    <link:loc xlink:href="http://xbrl.fasb.org/us-gaap/2019/elts/us-gaap-2019-01-31.xsd#us-gaap_AccumulatedDepreciationDepletionAndAmortizationPropertyPlantAndEquipment" xlink:label="loc_us-gaap_AccumulatedDepreciationDepletionAndAmortizationPropertyPlantAndEquipment_8E93F2D3893952A7A035AC78B1D7F650" xlink:type="locator" />
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    <link:label id="lab_us-gaap_PropertyPlantAndEquipmentNet_81D524CBAF849BC75E44E23266A6E5C9_totalLabel_en-US" xlink:label="lab_us-gaap_PropertyPlantAndEquipmentNet_C3B1A4AC0A3D5B128DD6549054A67D38" xlink:role="http://www.xbrl.org/2003/role/totalLabel" xlink:type="resource" xml:lang="en-US">Property and equipment, net</link:label>
    <link:loc xlink:href="http://xbrl.fasb.org/us-gaap/2019/elts/us-gaap-2019-01-31.xsd#us-gaap_PropertyPlantAndEquipmentNet" xlink:label="loc_us-gaap_PropertyPlantAndEquipmentNet_C3B1A4AC0A3D5B128DD6549054A67D38" xlink:type="locator" />
    <link:labelArc order="1" xlink:arcrole="http://www.xbrl.org/2003/arcrole/concept-label" xlink:from="loc_us-gaap_PropertyPlantAndEquipmentNet_C3B1A4AC0A3D5B128DD6549054A67D38" xlink:to="lab_us-gaap_PropertyPlantAndEquipmentNet_C3B1A4AC0A3D5B128DD6549054A67D38" xlink:type="arc" />
    <link:label id="lab_us-gaap_ShareBasedCompensationArrangementByShareBasedPaymentAwardOptionsOutstandingRollForward_DEC127E3012DBDD01C00E232662B53EA_terseLabel_en-US" xlink:label="lab_us-gaap_ShareBasedCompensationArrangementByShareBasedPaymentAwardOptionsOutstandingRollForward_B253E6E54EEE550DA26B2120752D018A" xlink:role="http://www.xbrl.org/2003/role/terseLabel" xlink:type="resource" xml:lang="en-US">Shares</link:label>
    <link:label id="lab_us-gaap_ShareBasedCompensationArrangementByShareBasedPaymentAwardOptionsOutstandingRollForward_DEC127E3012DBDD01C00E232662B53EA_label_en-US" xlink:label="lab_us-gaap_ShareBasedCompensationArrangementByShareBasedPaymentAwardOptionsOutstandingRollForward_B253E6E54EEE550DA26B2120752D018A" xlink:role="http://www.xbrl.org/2003/role/label" xlink:type="resource" xml:lang="en-US">Share-based Compensation Arrangement by Share-based Payment Award, Options, Outstanding [Roll Forward]</link:label>
    <link:loc xlink:href="http://xbrl.fasb.org/us-gaap/2019/elts/us-gaap-2019-01-31.xsd#us-gaap_ShareBasedCompensationArrangementByShareBasedPaymentAwardOptionsOutstandingRollForward" xlink:label="loc_us-gaap_ShareBasedCompensationArrangementByShareBasedPaymentAwardOptionsOutstandingRollForward_B253E6E54EEE550DA26B2120752D018A" xlink:type="locator" />
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    <link:label id="lab_us-gaap_ShareBasedCompensationArrangementByShareBasedPaymentAwardOptionsOutstandingNumber_C924C7CA6CC551777904E232662BEB24_periodStartLabel_en-US" xlink:label="lab_us-gaap_ShareBasedCompensationArrangementByShareBasedPaymentAwardOptionsOutstandingNumber_136142F19A6E5BA4B5092C01B7A7104F" xlink:role="http://www.xbrl.org/2003/role/periodStartLabel" xlink:type="resource" xml:lang="en-US">Options outstanding at beginning of period (in shares)</link:label>
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    <link:loc xlink:href="http://xbrl.fasb.org/us-gaap/2019/elts/us-gaap-2019-01-31.xsd#us-gaap_ShareBasedCompensationArrangementByShareBasedPaymentAwardOptionsOutstandingNumber" xlink:label="loc_us-gaap_ShareBasedCompensationArrangementByShareBasedPaymentAwardOptionsOutstandingNumber_136142F19A6E5BA4B5092C01B7A7104F" xlink:type="locator" />
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    <link:label id="lab_us-gaap_ShareBasedCompensationArrangementByShareBasedPaymentAwardOptionsGrantsInPeriodGross_1C1AC675E5E342B62FC4E232662C1CFF_terseLabel_en-US" xlink:label="lab_us-gaap_ShareBasedCompensationArrangementByShareBasedPaymentAwardOptionsGrantsInPeriodGross_36D54B8635C35155AE628C17C10B66D1" xlink:role="http://www.xbrl.org/2003/role/terseLabel" xlink:type="resource" xml:lang="en-US">Granted (in shares)</link:label>
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    <link:loc xlink:href="http://xbrl.fasb.org/us-gaap/2019/elts/us-gaap-2019-01-31.xsd#us-gaap_ShareBasedCompensationArrangementByShareBasedPaymentAwardOptionsGrantsInPeriodGross" xlink:label="loc_us-gaap_ShareBasedCompensationArrangementByShareBasedPaymentAwardOptionsGrantsInPeriodGross_36D54B8635C35155AE628C17C10B66D1" xlink:type="locator" />
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    <link:loc xlink:href="http://xbrl.fasb.org/us-gaap/2019/elts/us-gaap-2019-01-31.xsd#us-gaap_ShareBasedCompensationArrangementByShareBasedPaymentAwardOptionsForfeituresInPeriod" xlink:label="loc_us-gaap_ShareBasedCompensationArrangementByShareBasedPaymentAwardOptionsForfeituresInPeriod_41260A25DEAD52E9B5ED8BD90C183E64" xlink:type="locator" />
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    <link:label id="lab_exel_LesseeOperatingLeaseLiabilityTenantImprovementReimbursements_A9B94EE88334E9B3F10A0F9CE28C8D53_terseLabel_en-US" xlink:label="lab_exel_LesseeOperatingLeaseLiabilityTenantImprovementReimbursements_A9B94EE88334E9B3F10A0F9CE28C8D53" xlink:role="http://www.xbrl.org/2003/role/terseLabel" xlink:type="resource" xml:lang="en-US">Tenant improvement reimbursements</link:label>
    <link:label id="lab_exel_LesseeOperatingLeaseLiabilityTenantImprovementReimbursements_A9B94EE88334E9B3F10A0F9CE28C8D53_label_en-US" xlink:label="lab_exel_LesseeOperatingLeaseLiabilityTenantImprovementReimbursements_A9B94EE88334E9B3F10A0F9CE28C8D53" xlink:role="http://www.xbrl.org/2003/role/label" xlink:type="resource" xml:lang="en-US">Lessee, Operating Lease, Liability, Tenant Improvement Reimbursements</link:label>
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    <link:loc xlink:href="exel-20190927.xsd#exel_LesseeOperatingLeaseLiabilityTenantImprovementReimbursements" xlink:label="loc_exel_LesseeOperatingLeaseLiabilityTenantImprovementReimbursements_A9B94EE88334E9B3F10A0F9CE28C8D53" xlink:type="locator" />
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    <link:label id="lab_exel_OperatingLeaseSurrenderedAreaOfRealEstateProperty_D874D8CE9A44B0BDD8820F9CE28D47DC_terseLabel_en-US" xlink:label="lab_exel_OperatingLeaseSurrenderedAreaOfRealEstateProperty_D874D8CE9A44B0BDD8820F9CE28D47DC" xlink:role="http://www.xbrl.org/2003/role/terseLabel" xlink:type="resource" xml:lang="en-US">Operating lease, surrendered (in square feet)</link:label>
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    <link:label id="lab_exel_ProductGrossMember_80DDD285E2BD09A5DA97B3E452349752_label_en-US" xlink:label="lab_exel_ProductGrossMember_80DDD285E2BD09A5DA97B3E452349752" xlink:role="http://www.xbrl.org/2003/role/label" xlink:type="resource" xml:lang="en-US">Product, Gross [Member]</link:label>
    <link:label id="lab_exel_ProductGrossMember_80DDD285E2BD09A5DA97B3E452349752_documentation_en-US" xlink:label="lab_exel_ProductGrossMember_80DDD285E2BD09A5DA97B3E452349752" xlink:role="http://www.xbrl.org/2003/role/documentation" xlink:type="resource" xml:lang="en-US">Product, Gross [Member]</link:label>
    <link:loc xlink:href="exel-20190927.xsd#exel_ProductGrossMember" xlink:label="loc_exel_ProductGrossMember_80DDD285E2BD09A5DA97B3E452349752" xlink:type="locator" />
    <link:labelArc order="1" xlink:arcrole="http://www.xbrl.org/2003/arcrole/concept-label" xlink:from="loc_exel_ProductGrossMember_80DDD285E2BD09A5DA97B3E452349752" xlink:to="lab_exel_ProductGrossMember_80DDD285E2BD09A5DA97B3E452349752" xlink:type="arc" />
    <link:label id="lab_exel_SalesDiscountsAndAllowancesMember_3CA16FBD297A6C682B1BB3E45234A7B8_terseLabel_en-US" xlink:label="lab_exel_SalesDiscountsAndAllowancesMember_3CA16FBD297A6C682B1BB3E45234A7B8" xlink:role="http://www.xbrl.org/2003/role/terseLabel" xlink:type="resource" xml:lang="en-US">Discounts and allowances</link:label>
    <link:label id="lab_exel_SalesDiscountsAndAllowancesMember_3CA16FBD297A6C682B1BB3E45234A7B8_label_en-US" xlink:label="lab_exel_SalesDiscountsAndAllowancesMember_3CA16FBD297A6C682B1BB3E45234A7B8" xlink:role="http://www.xbrl.org/2003/role/label" xlink:type="resource" xml:lang="en-US">Sales Discounts And Allowances [Member]</link:label>
    <link:label id="lab_exel_SalesDiscountsAndAllowancesMember_3CA16FBD297A6C682B1BB3E45234A7B8_documentation_en-US" xlink:label="lab_exel_SalesDiscountsAndAllowancesMember_3CA16FBD297A6C682B1BB3E45234A7B8" xlink:role="http://www.xbrl.org/2003/role/documentation" xlink:type="resource" xml:lang="en-US">Sales Discounts And Allowances [Member]</link:label>
    <link:loc xlink:href="exel-20190927.xsd#exel_SalesDiscountsAndAllowancesMember" xlink:label="loc_exel_SalesDiscountsAndAllowancesMember_3CA16FBD297A6C682B1BB3E45234A7B8" xlink:type="locator" />
    <link:labelArc order="1" xlink:arcrole="http://www.xbrl.org/2003/arcrole/concept-label" xlink:from="loc_exel_SalesDiscountsAndAllowancesMember_3CA16FBD297A6C682B1BB3E45234A7B8" xlink:to="lab_exel_SalesDiscountsAndAllowancesMember_3CA16FBD297A6C682B1BB3E45234A7B8" xlink:type="arc" />
    <link:label id="lab_exel_CollaborationMember_95878F4B06C57133FFA0B3E45235B517_verboseLabel_en-US" xlink:label="lab_exel_CollaborationMember_95878F4B06C57133FFA0B3E45235B517" xlink:role="http://www.xbrl.org/2003/role/verboseLabel" xlink:type="resource" xml:lang="en-US">Total collaboration revenues</link:label>
    <link:loc xlink:href="exel-20190927.xsd#exel_CollaborationMember" xlink:label="loc_exel_CollaborationMember_95878F4B06C57133FFA0B3E45235B517" xlink:type="locator" />
    <link:labelArc order="1" xlink:arcrole="http://www.xbrl.org/2003/arcrole/concept-label" xlink:from="loc_exel_CollaborationMember_95878F4B06C57133FFA0B3E45235B517" xlink:to="lab_exel_CollaborationMember_95878F4B06C57133FFA0B3E45235B517" xlink:type="arc" />
    <link:label id="lab_us-gaap_LicenseMember_F60C673DDA19211FAF7DB3E452354945_verboseLabel_en-US" xlink:label="lab_us-gaap_LicenseMember_F60C673DDA19211FAF7DB3E452354945" xlink:role="http://www.xbrl.org/2003/role/verboseLabel" xlink:type="resource" xml:lang="en-US">License revenues</link:label>
    <link:label id="lab_us-gaap_LicenseMember_F60C673DDA19211FAF7DB3E452354945_label_en-US" xlink:label="lab_us-gaap_LicenseMember_F60C673DDA19211FAF7DB3E452354945" xlink:role="http://www.xbrl.org/2003/role/label" xlink:type="resource" xml:lang="en-US">License [Member]</link:label>
    <link:loc xlink:href="http://xbrl.fasb.org/us-gaap/2019/elts/us-gaap-2019-01-31.xsd#us-gaap_LicenseMember" xlink:label="loc_us-gaap_LicenseMember_F60C673DDA19211FAF7DB3E452354945" xlink:type="locator" />
    <link:labelArc order="1" xlink:arcrole="http://www.xbrl.org/2003/arcrole/concept-label" xlink:from="loc_us-gaap_LicenseMember_F60C673DDA19211FAF7DB3E452354945" xlink:to="lab_us-gaap_LicenseMember_F60C673DDA19211FAF7DB3E452354945" xlink:type="arc" />
    <link:label id="lab_exel_ResearchandDevelopmentMember_A3D7509907FAA8F8088BB3E452355D2D_terseLabel_en-US" xlink:label="lab_exel_ResearchandDevelopmentMember_A3D7509907FAA8F8088BB3E452355D2D" xlink:role="http://www.xbrl.org/2003/role/terseLabel" xlink:type="resource" xml:lang="en-US">Research and development services revenues</link:label>
    <link:label id="lab_exel_ResearchandDevelopmentMember_A3D7509907FAA8F8088BB3E452355D2D_label_en-US" xlink:label="lab_exel_ResearchandDevelopmentMember_A3D7509907FAA8F8088BB3E452355D2D" xlink:role="http://www.xbrl.org/2003/role/label" xlink:type="resource" xml:lang="en-US">Research and Development [Member]</link:label>
    <link:label id="lab_exel_ResearchandDevelopmentMember_A3D7509907FAA8F8088BB3E452355D2D_documentation_en-US" xlink:label="lab_exel_ResearchandDevelopmentMember_A3D7509907FAA8F8088BB3E452355D2D" xlink:role="http://www.xbrl.org/2003/role/documentation" xlink:type="resource" xml:lang="en-US">Research and Development [Member]</link:label>
    <link:loc xlink:href="exel-20190927.xsd#exel_ResearchandDevelopmentMember" xlink:label="loc_exel_ResearchandDevelopmentMember_A3D7509907FAA8F8088BB3E452355D2D" xlink:type="locator" />
    <link:labelArc order="1" xlink:arcrole="http://www.xbrl.org/2003/arcrole/concept-label" xlink:from="loc_exel_ResearchandDevelopmentMember_A3D7509907FAA8F8088BB3E452355D2D" xlink:to="lab_exel_ResearchandDevelopmentMember_A3D7509907FAA8F8088BB3E452355D2D" xlink:type="arc" />
    <link:label id="lab_exel_OtherCollaborationMember_5C4582BF1FCFEA54E7DCB3E45235608D_terseLabel_en-US" xlink:label="lab_exel_OtherCollaborationMember_5C4582BF1FCFEA54E7DCB3E45235608D" xlink:role="http://www.xbrl.org/2003/role/terseLabel" xlink:type="resource" xml:lang="en-US">Other collaboration revenues</link:label>
    <link:label id="lab_exel_OtherCollaborationMember_5C4582BF1FCFEA54E7DCB3E45235608D_label_en-US" xlink:label="lab_exel_OtherCollaborationMember_5C4582BF1FCFEA54E7DCB3E45235608D" xlink:role="http://www.xbrl.org/2003/role/label" xlink:type="resource" xml:lang="en-US">Other Collaboration [Member]</link:label>
    <link:label id="lab_exel_OtherCollaborationMember_5C4582BF1FCFEA54E7DCB3E45235608D_documentation_en-US" xlink:label="lab_exel_OtherCollaborationMember_5C4582BF1FCFEA54E7DCB3E45235608D" xlink:role="http://www.xbrl.org/2003/role/documentation" xlink:type="resource" xml:lang="en-US">Other Collaboration [Member]</link:label>
    <link:loc xlink:href="exel-20190927.xsd#exel_OtherCollaborationMember" xlink:label="loc_exel_OtherCollaborationMember_5C4582BF1FCFEA54E7DCB3E45235608D" xlink:type="locator" />
    <link:labelArc order="1" xlink:arcrole="http://www.xbrl.org/2003/arcrole/concept-label" xlink:from="loc_exel_OtherCollaborationMember_5C4582BF1FCFEA54E7DCB3E45235608D" xlink:to="lab_exel_OtherCollaborationMember_5C4582BF1FCFEA54E7DCB3E45235608D" xlink:type="arc" />
    <link:label id="lab_us-gaap_OperatingLeaseLiabilitiesPaymentsDueAbstract_24169C126C7CBFB890300F844C3C0909_terseLabel_en-US" xlink:label="lab_us-gaap_OperatingLeaseLiabilitiesPaymentsDueAbstract_24169C126C7CBFB890300F844C3C0909" xlink:role="http://www.xbrl.org/2003/role/terseLabel" xlink:type="resource" xml:lang="en-US">Maturities of Operating Lease Liabilities</link:label>
    <link:label id="lab_us-gaap_OperatingLeaseLiabilitiesPaymentsDueAbstract_24169C126C7CBFB890300F844C3C0909_label_en-US" xlink:label="lab_us-gaap_OperatingLeaseLiabilitiesPaymentsDueAbstract_24169C126C7CBFB890300F844C3C0909" xlink:role="http://www.xbrl.org/2003/role/label" xlink:type="resource" xml:lang="en-US">Lessee, Operating Lease, Liability, Payment, Due [Abstract]</link:label>
    <link:loc xlink:href="http://xbrl.fasb.org/us-gaap/2019/elts/us-gaap-2019-01-31.xsd#us-gaap_OperatingLeaseLiabilitiesPaymentsDueAbstract" xlink:label="loc_us-gaap_OperatingLeaseLiabilitiesPaymentsDueAbstract_24169C126C7CBFB890300F844C3C0909" xlink:type="locator" />
    <link:labelArc order="1" xlink:arcrole="http://www.xbrl.org/2003/arcrole/concept-label" xlink:from="loc_us-gaap_OperatingLeaseLiabilitiesPaymentsDueAbstract_24169C126C7CBFB890300F844C3C0909" xlink:to="lab_us-gaap_OperatingLeaseLiabilitiesPaymentsDueAbstract_24169C126C7CBFB890300F844C3C0909" xlink:type="arc" />
    <link:label id="lab_us-gaap_LesseeOperatingLeaseLiabilityPaymentsRemainderOfFiscalYear_350A5742ABB7CF7C95FF0F844C3C3B80_terseLabel_en-US" xlink:label="lab_us-gaap_LesseeOperatingLeaseLiabilityPaymentsRemainderOfFiscalYear_350A5742ABB7CF7C95FF0F844C3C3B80" xlink:role="http://www.xbrl.org/2003/role/terseLabel" xlink:type="resource" xml:lang="en-US">Remainder of 2019</link:label>
    <link:label id="lab_us-gaap_LesseeOperatingLeaseLiabilityPaymentsRemainderOfFiscalYear_350A5742ABB7CF7C95FF0F844C3C3B80_label_en-US" xlink:label="lab_us-gaap_LesseeOperatingLeaseLiabilityPaymentsRemainderOfFiscalYear_350A5742ABB7CF7C95FF0F844C3C3B80" xlink:role="http://www.xbrl.org/2003/role/label" xlink:type="resource" xml:lang="en-US">Lessee, Operating Lease, Liability, Payments, Remainder of Fiscal Year</link:label>
    <link:loc xlink:href="http://xbrl.fasb.org/us-gaap/2019/elts/us-gaap-2019-01-31.xsd#us-gaap_LesseeOperatingLeaseLiabilityPaymentsRemainderOfFiscalYear" xlink:label="loc_us-gaap_LesseeOperatingLeaseLiabilityPaymentsRemainderOfFiscalYear_350A5742ABB7CF7C95FF0F844C3C3B80" xlink:type="locator" />
    <link:labelArc order="1" xlink:arcrole="http://www.xbrl.org/2003/arcrole/concept-label" xlink:from="loc_us-gaap_LesseeOperatingLeaseLiabilityPaymentsRemainderOfFiscalYear_350A5742ABB7CF7C95FF0F844C3C3B80" xlink:to="lab_us-gaap_LesseeOperatingLeaseLiabilityPaymentsRemainderOfFiscalYear_350A5742ABB7CF7C95FF0F844C3C3B80" xlink:type="arc" />
    <link:label id="lab_exel_OperatingLeaseLiabilitiesDurationOfMaturityAbstract_87CDD4D6BD02DED907D60F844C3DB3E4_terseLabel_en-US" xlink:label="lab_exel_OperatingLeaseLiabilitiesDurationOfMaturityAbstract_87CDD4D6BD02DED907D60F844C3DB3E4" xlink:role="http://www.xbrl.org/2003/role/terseLabel" xlink:type="resource" xml:lang="en-US">Years ending December 31,</link:label>
    <link:label id="lab_exel_OperatingLeaseLiabilitiesDurationOfMaturityAbstract_87CDD4D6BD02DED907D60F844C3DB3E4_label_en-US" xlink:label="lab_exel_OperatingLeaseLiabilitiesDurationOfMaturityAbstract_87CDD4D6BD02DED907D60F844C3DB3E4" xlink:role="http://www.xbrl.org/2003/role/label" xlink:type="resource" xml:lang="en-US">Operating Lease Liabilities, Duration Of Maturity [Abstract]</link:label>
    <link:label id="lab_exel_OperatingLeaseLiabilitiesDurationOfMaturityAbstract_87CDD4D6BD02DED907D60F844C3DB3E4_documentation_en-US" xlink:label="lab_exel_OperatingLeaseLiabilitiesDurationOfMaturityAbstract_87CDD4D6BD02DED907D60F844C3DB3E4" xlink:role="http://www.xbrl.org/2003/role/documentation" xlink:type="resource" xml:lang="en-US">Operating Lease Liabilities, Duration Of Maturity [Abstract]</link:label>
    <link:loc xlink:href="exel-20190927.xsd#exel_OperatingLeaseLiabilitiesDurationOfMaturityAbstract" xlink:label="loc_exel_OperatingLeaseLiabilitiesDurationOfMaturityAbstract_87CDD4D6BD02DED907D60F844C3DB3E4" xlink:type="locator" />
    <link:labelArc order="1" xlink:arcrole="http://www.xbrl.org/2003/arcrole/concept-label" xlink:from="loc_exel_OperatingLeaseLiabilitiesDurationOfMaturityAbstract_87CDD4D6BD02DED907D60F844C3DB3E4" xlink:to="lab_exel_OperatingLeaseLiabilitiesDurationOfMaturityAbstract_87CDD4D6BD02DED907D60F844C3DB3E4" xlink:type="arc" />
    <link:label id="lab_us-gaap_LesseeOperatingLeaseLiabilityPaymentsDueYearTwo_88481A79624731142CBF0F844C3D2416_terseLabel_en-US" xlink:label="lab_us-gaap_LesseeOperatingLeaseLiabilityPaymentsDueYearTwo_88481A79624731142CBF0F844C3D2416" xlink:role="http://www.xbrl.org/2003/role/terseLabel" xlink:type="resource" xml:lang="en-US">2020</link:label>
    <link:label id="lab_us-gaap_LesseeOperatingLeaseLiabilityPaymentsDueYearTwo_88481A79624731142CBF0F844C3D2416_label_en-US" xlink:label="lab_us-gaap_LesseeOperatingLeaseLiabilityPaymentsDueYearTwo_88481A79624731142CBF0F844C3D2416" xlink:role="http://www.xbrl.org/2003/role/label" xlink:type="resource" xml:lang="en-US">Lessee, Operating Lease, Liability, Payments, Due Year Two</link:label>
    <link:loc xlink:href="http://xbrl.fasb.org/us-gaap/2019/elts/us-gaap-2019-01-31.xsd#us-gaap_LesseeOperatingLeaseLiabilityPaymentsDueYearTwo" xlink:label="loc_us-gaap_LesseeOperatingLeaseLiabilityPaymentsDueYearTwo_88481A79624731142CBF0F844C3D2416" xlink:type="locator" />
    <link:labelArc order="1" xlink:arcrole="http://www.xbrl.org/2003/arcrole/concept-label" xlink:from="loc_us-gaap_LesseeOperatingLeaseLiabilityPaymentsDueYearTwo_88481A79624731142CBF0F844C3D2416" xlink:to="lab_us-gaap_LesseeOperatingLeaseLiabilityPaymentsDueYearTwo_88481A79624731142CBF0F844C3D2416" xlink:type="arc" />
    <link:label id="lab_us-gaap_LesseeOperatingLeaseLiabilityPaymentsDueYearThree_F40271ED025AE9FAC35A0F844C3EAF04_terseLabel_en-US" xlink:label="lab_us-gaap_LesseeOperatingLeaseLiabilityPaymentsDueYearThree_F40271ED025AE9FAC35A0F844C3EAF04" xlink:role="http://www.xbrl.org/2003/role/terseLabel" xlink:type="resource" xml:lang="en-US">2021</link:label>
    <link:label id="lab_us-gaap_LesseeOperatingLeaseLiabilityPaymentsDueYearThree_F40271ED025AE9FAC35A0F844C3EAF04_label_en-US" xlink:label="lab_us-gaap_LesseeOperatingLeaseLiabilityPaymentsDueYearThree_F40271ED025AE9FAC35A0F844C3EAF04" xlink:role="http://www.xbrl.org/2003/role/label" xlink:type="resource" xml:lang="en-US">Lessee, Operating Lease, Liability, Payments, Due Year Three</link:label>
    <link:loc xlink:href="http://xbrl.fasb.org/us-gaap/2019/elts/us-gaap-2019-01-31.xsd#us-gaap_LesseeOperatingLeaseLiabilityPaymentsDueYearThree" xlink:label="loc_us-gaap_LesseeOperatingLeaseLiabilityPaymentsDueYearThree_F40271ED025AE9FAC35A0F844C3EAF04" xlink:type="locator" />
    <link:labelArc order="1" xlink:arcrole="http://www.xbrl.org/2003/arcrole/concept-label" xlink:from="loc_us-gaap_LesseeOperatingLeaseLiabilityPaymentsDueYearThree_F40271ED025AE9FAC35A0F844C3EAF04" xlink:to="lab_us-gaap_LesseeOperatingLeaseLiabilityPaymentsDueYearThree_F40271ED025AE9FAC35A0F844C3EAF04" xlink:type="arc" />
    <link:label id="lab_us-gaap_LesseeOperatingLeaseLiabilityPaymentsDueYearFour_47A53C0562B19B830E830F844C3EAD7F_terseLabel_en-US" xlink:label="lab_us-gaap_LesseeOperatingLeaseLiabilityPaymentsDueYearFour_47A53C0562B19B830E830F844C3EAD7F" xlink:role="http://www.xbrl.org/2003/role/terseLabel" xlink:type="resource" xml:lang="en-US">2022</link:label>
    <link:label id="lab_us-gaap_LesseeOperatingLeaseLiabilityPaymentsDueYearFour_47A53C0562B19B830E830F844C3EAD7F_label_en-US" xlink:label="lab_us-gaap_LesseeOperatingLeaseLiabilityPaymentsDueYearFour_47A53C0562B19B830E830F844C3EAD7F" xlink:role="http://www.xbrl.org/2003/role/label" xlink:type="resource" xml:lang="en-US">Lessee, Operating Lease, Liability, Payments, Due Year Four</link:label>
    <link:loc xlink:href="http://xbrl.fasb.org/us-gaap/2019/elts/us-gaap-2019-01-31.xsd#us-gaap_LesseeOperatingLeaseLiabilityPaymentsDueYearFour" xlink:label="loc_us-gaap_LesseeOperatingLeaseLiabilityPaymentsDueYearFour_47A53C0562B19B830E830F844C3EAD7F" xlink:type="locator" />
    <link:labelArc order="1" xlink:arcrole="http://www.xbrl.org/2003/arcrole/concept-label" xlink:from="loc_us-gaap_LesseeOperatingLeaseLiabilityPaymentsDueYearFour_47A53C0562B19B830E830F844C3EAD7F" xlink:to="lab_us-gaap_LesseeOperatingLeaseLiabilityPaymentsDueYearFour_47A53C0562B19B830E830F844C3EAD7F" xlink:type="arc" />
    <link:label id="lab_us-gaap_LesseeOperatingLeaseLiabilityPaymentsDueYearFive_9909FD86871D5BDEBF9C0F844C3E8A7B_terseLabel_en-US" xlink:label="lab_us-gaap_LesseeOperatingLeaseLiabilityPaymentsDueYearFive_9909FD86871D5BDEBF9C0F844C3E8A7B" xlink:role="http://www.xbrl.org/2003/role/terseLabel" xlink:type="resource" xml:lang="en-US">2023</link:label>
    <link:label id="lab_us-gaap_LesseeOperatingLeaseLiabilityPaymentsDueYearFive_9909FD86871D5BDEBF9C0F844C3E8A7B_label_en-US" xlink:label="lab_us-gaap_LesseeOperatingLeaseLiabilityPaymentsDueYearFive_9909FD86871D5BDEBF9C0F844C3E8A7B" xlink:role="http://www.xbrl.org/2003/role/label" xlink:type="resource" xml:lang="en-US">Lessee, Operating Lease, Liability, Payments, Due Year Five</link:label>
    <link:loc xlink:href="http://xbrl.fasb.org/us-gaap/2019/elts/us-gaap-2019-01-31.xsd#us-gaap_LesseeOperatingLeaseLiabilityPaymentsDueYearFive" xlink:label="loc_us-gaap_LesseeOperatingLeaseLiabilityPaymentsDueYearFive_9909FD86871D5BDEBF9C0F844C3E8A7B" xlink:type="locator" />
    <link:labelArc order="1" xlink:arcrole="http://www.xbrl.org/2003/arcrole/concept-label" xlink:from="loc_us-gaap_LesseeOperatingLeaseLiabilityPaymentsDueYearFive_9909FD86871D5BDEBF9C0F844C3E8A7B" xlink:to="lab_us-gaap_LesseeOperatingLeaseLiabilityPaymentsDueYearFive_9909FD86871D5BDEBF9C0F844C3E8A7B" xlink:type="arc" />
    <link:label id="lab_us-gaap_LesseeOperatingLeaseLiabilityPaymentsDueAfterYearFive_8430FB11B858A63A20010F844C3E1945_terseLabel_en-US" xlink:label="lab_us-gaap_LesseeOperatingLeaseLiabilityPaymentsDueAfterYearFive_8430FB11B858A63A20010F844C3E1945" xlink:role="http://www.xbrl.org/2003/role/terseLabel" xlink:type="resource" xml:lang="en-US">Thereafter</link:label>
    <link:label id="lab_us-gaap_LesseeOperatingLeaseLiabilityPaymentsDueAfterYearFive_8430FB11B858A63A20010F844C3E1945_label_en-US" xlink:label="lab_us-gaap_LesseeOperatingLeaseLiabilityPaymentsDueAfterYearFive_8430FB11B858A63A20010F844C3E1945" xlink:role="http://www.xbrl.org/2003/role/label" xlink:type="resource" xml:lang="en-US">Lessee, Operating Lease, Liability, Payments, Due after Year Five</link:label>
    <link:loc xlink:href="http://xbrl.fasb.org/us-gaap/2019/elts/us-gaap-2019-01-31.xsd#us-gaap_LesseeOperatingLeaseLiabilityPaymentsDueAfterYearFive" xlink:label="loc_us-gaap_LesseeOperatingLeaseLiabilityPaymentsDueAfterYearFive_8430FB11B858A63A20010F844C3E1945" xlink:type="locator" />
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